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P28347 | TEAD1_HUMAN | Transcriptional enhancer factor TEF-1 (TEAD1)
3D structures mapped by conservation among orthologs
[ Domain: "tri-helical" // TEA ]
2HZD
4Z8E
5NNX
download pymol session
[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // KOG3841 ]
3KYS
4RE1
6HIL
6IM5
download pymol session
[ Alpha Fold Model ]
(go)
Known binders annotated in ChEMBL
IC50 table
molecule_chembl_id
structure
assay_type
relation
values
units
mol_wt
smiles
organism
assay_chembl_id
bao_label
CHEMBL4129172
OBDepict
O
NH
S
N
N
N
H
IC50
=
83.0
nM
368.51
O=C(CSc1nnc[nH]1)Nc1ccc(C2C3CC4CC(C3)CC2C4)cc1
Homo sapiens
CHEMBL4120897
cell-based format