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Q460N3 | PAR15_HUMAN | Protein mono-ADP-ribosyltransferase PARP15 (PARP15)
3D structures mapped by conservation among orthologs
[ Domain: "ADP-ribosylation" // PARP ]
3BLJ
3GEY
4F0E
6EK3
download pymol session
[ Domain: "Macro domain-like" // Macro ]
3V2B
download pymol session
[ Alpha Fold Model ]
(go)
Known binders annotated in ChEMBL
IC50 table
molecule_chembl_id
structure
assay_type
relation
values
units
mol_wt
smiles
organism
assay_chembl_id
bao_label
CHEMBL4089522
OBDepict
O
NH
N
O
O
NH
2
N
F
IC50
=
520.0
nM
396.42
NC(=O)c1cccc(NC(=O)/C=CC(=O)N2CCN(c3ccc(F)cc3)CC2)c1
Homo sapiens
CHEMBL4022069
single protein format