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Q86U86 | PB1_HUMAN | Protein polybromo-1 (PBRM1)
3D structures mapped by conservation among orthologs
[ Domain: "Bromodomain" // Bromodomain ]
2KTB
3G0J
3HMF
3IU5
3IU6
3K2J
3LJW
3MB4
3TLP
4Q0N
4Q0O
4Y03
5E7D
5FH6
5FH7
5FH8
5HRV
5HRW
5HRX
5II1
5II2
5IID
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[ Alpha Fold Model ]
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Known binders annotated in ChEMBL
IC50 table
molecule_chembl_id
structure
assay_type
relation
values
units
mol_wt
smiles
organism
assay_chembl_id
bao_label
CHEMBL4650213
OBDepict
O
HO
N
H
H
N
N
IC50
=
550.3
nM
321.38
O=C(C=CN1C[C@H]2C[C@@H]1CN2c1ccccn1)c1ccccc1O
Homo sapiens
CHEMBL4650019
single protein format