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Q8N5Y8 | PAR16_HUMAN | Protein mono-ADP-ribosyltransferase PARP16 (PARP16)
3D structures mapped by conservation among orthologs
[ Domain: "ADP-ribosylation" // PARP ]
4F0D
6HXR
6HXS
download pymol session
[ Domain: "Domain of poly(ADP-ribose) polymerase" // EUF08131 ]
4F0D
6HXR
6HXS
download pymol session
[ Domain: pdbs with more than 2 multi-domains ]
6HXR
download pymol session
[ Alpha Fold Model ]
(go)
Known binders annotated in ChEMBL
IC50 table
molecule_chembl_id
structure
assay_type
relation
values
units
mol_wt
smiles
organism
assay_chembl_id
bao_label
CHEMBL4089522
OBDepict
O
NH
N
O
O
NH
2
N
F
IC50
=
560.0
nM
396.42
NC(=O)c1cccc(NC(=O)/C=CC(=O)N2CCN(c3ccc(F)cc3)CC2)c1
Homo sapiens
CHEMBL4022070
single protein format