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Q92830 | KAT2A_HUMAN | Histone acetyltransferase KAT2A (KAT2A)
3D structures mapped by conservation among orthologs
[ Domain: "Acyl-CoA N-acyltransferases (Nat)" // Acetyltransf_10 ]
1Z4R
5H84
5H86
5TRL
5TRM
download pymol session
[ Domain: "Bromodomain" // Bromodomain ]
1F68
3D7C
5MLJ
6J3P
download pymol session
[ Domain: pdbs with more than 2 multi-domains ]
5TRL
5TRM
download pymol session
[ Alpha Fold Model ]
(go)
Known binders annotated in ChEMBL
Ki table
molecule_chembl_id
structure
assay_type
relation
values
units
mol_wt
smiles
organism
assay_chembl_id
bao_label
CHEMBL4069412
OBDepict
CH
3
N
H
N
H
H
N
Br
N
O
CH
3
Ki
=
1.4
nM
377.29
CN1C[C@H](Nc2cnn(C)c(=O)c2Br)C[C@H](c2ccccc2)C1
Homo sapiens
CHEMBL4003548
assay format