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Q9NZN5 | ARHGC_HUMAN | Rho guanine nucleotide exchange factor 12 (ARHGEF12)
3D structures mapped by conservation among orthologs
[ Domain: "DBL homology domain (DH-domain)" // RhoGEF ]
1TXD
1X86
download pymol session
[ Domain: "PH domain-like" // PH_13_1 ]
1TXD
1X86
download pymol session
[ Domain: "PDZ domain" // PDZ ]
2OMJ
2OS6
download pymol session
[ Alpha Fold Model ]
(go)
Known binders annotated in ChEMBL
IC50 table
molecule_chembl_id
structure
assay_type
relation
values
units
mol_wt
smiles
organism
assay_chembl_id
bao_label
CHEMBL485210
OBDepict
CH
3
O
O
N
H
O
N
IC50
=
1000.0
nM
384.44
Cc1cccc(COc2cccc(/C=C3C(=O)NN(c4ccccc4)C3=O)c2)c1
Homo sapiens
CHEMBL4419711
single protein format